Table 2.

Cutoff values for in vitro hazard profiling.

No responseWeak responseStrong response
Receptor activity assaysNo responseEC10 or IC10 > 5 μMEC10 or IC10 < 5 μM
TTR bindingNo responseEC10 or IC10 > 100 nMEC10 or IC10 < 100 nM
H295RNo responseECIR1.5 > 2 μMECIR1.5 < 2 μM
No responseWeak responseStrong response
Receptor activity assaysNo responseEC10 or IC10 > 5 μMEC10 or IC10 < 5 μM
TTR bindingNo responseEC10 or IC10 > 100 nMEC10 or IC10 < 100 nM
H295RNo responseECIR1.5 > 2 μMECIR1.5 < 2 μM
Table 2.

Cutoff values for in vitro hazard profiling.

No responseWeak responseStrong response
Receptor activity assaysNo responseEC10 or IC10 > 5 μMEC10 or IC10 < 5 μM
TTR bindingNo responseEC10 or IC10 > 100 nMEC10 or IC10 < 100 nM
H295RNo responseECIR1.5 > 2 μMECIR1.5 < 2 μM
No responseWeak responseStrong response
Receptor activity assaysNo responseEC10 or IC10 > 5 μMEC10 or IC10 < 5 μM
TTR bindingNo responseEC10 or IC10 > 100 nMEC10 or IC10 < 100 nM
H295RNo responseECIR1.5 > 2 μMECIR1.5 < 2 μM
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